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Tocris/L Moses dihydrochloride/6251/50/50 mg
  • Tocris/L Moses dihydrochloride/6251/50/50 mg

Tocris/L Moses dihydrochloride/6251/50/50 mg

价格: ¥7548.00 市场价: 12580.00

货号: 6251/50
品牌: Tocris
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    • Description:HighaffinityandselectivePCAFbromodomaininhibitor
      ChemicalName:(1S,2S)-N1,N1-Dimethyl-N2-(3-methyl-1,2,4-triazolo[3,4-a]phthalazin-6-yl)-1-phenylpropane-1,2-diaminedihydrochloride
      Purity:≥98%(HPLC)
      BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

      BiologicalActivity

      Highaffinityandselectivecell-permeablep300/CBP-associatedfactor(PCAF)inhibitor(Ki=47nM).Exhibitsnosignificantactivityagainstapanelof48otherbromodomainsexceptGCN5(Kd=600nM).Exhibits>4500-foldselectivityforPCAFoverBRD4.AlsoexhibitsmetabolicstABIlityinmouseandhumanlivermicrosomesandnoobservablecytotoxicityinperipheralbloodmononuclearcells(PBMC).

      LicensingInformation

      ThiscompoundissuppliedinconjunctionwiththeStructuralGenomicsConsortium.Forfurthercharacterizationdetails,pleasevisittheL-MosesprobesummaryontheSGCwebsite.

      TechnicalData

      M.Wt433.38
      FormulaC21H24N6.2HCl
      StorageDesiccateatRT
      Purity≥98%(HPLC)
      SmilesC[C@@H]([C@H](C1=CC=CC=C1)N(C)C)NC2=NN3C(C)=NN=C3C4=CC=CC=C24

      Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

      AllTocrisproductsareintendedforlaboratoryresearchuseonly.

      SolubilityData

      SolubilitySolubleto100mMinwaterandto100mMinDMSO

      PreparingStockSolutions

      Thefollowingdataisbasedontheproductmolecularweight433.38.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

      Concentration/SolventVolume/Mass1mg5mg10mg
      1mM2.31mL11.54mL23.07mL
      5mM0.46mL2.31mL4.61mL
      10mM0.23mL1.15mL2.31mL
      50mM0.05mL0.23mL0.46mL

      ProductDatasheets

      CertificateofAnalysis/ProductDatasheet
      SafetyDatasheet

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