当前位置 ： Tocris >>> Tocris/TASP 0390325/5729/10/10 mg
Tocris/TASP 0390325/5729/10/10 mg
  • Tocris/TASP 0390325/5729/10/10 mg

Tocris/TASP 0390325/5729/10/10 mg

价格: ¥2388.00 市场价: 3980.00
打印产品信息
货号: 5729
品牌: Tocris
规格
数量
库存(0)
特别 提示
代购产品：无质量问题不接受退换货，下单前请仔细核对信息。
下单后请及时联系客服核对商品价格，订单生效后再付款。
立即购买 加入购物车

收藏商品
资深产品顾问
咨询顾问

全国免费服务热线

4000-520-616

  • 自营商城 一站式服务
  • 厂家直采 剔除溢价
  • 品质甄选 正品保证
  • 严控流程 只做188精品
  • 极速物流 如约送货
  • 详情
  • 使用说明
  • 常见问题
    • Description:PotentandselectiveV1BreceptorantagoNIST;orallybioavailable
      ChemicalName:2-(3-Chloro-4-fluorophenyl)-N-(1-methylethyl)-6-[3-(4-morpholinyl)propoxy]-4-oxo-pyrido[2,3-d]pyrimidine-3(4H)-acetamidehydrochloride
      Purity:≥98%(HPLC)
      BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

      BiologicalActivity

      PotentandselectiveV1Breceptorantagonist(IC50=2.22nMforratpituitaryreceptor).Exhibitsnosignificantaffinityfor85otherreceptors,ionchannelsandtransportersat10μM,includingV1AandV2.IncreasesACTHlevelsinrats.Orallybioavailable.Antidepressantandanxiolytic.

      TechnicalData

      M.Wt554.44
      FormulaC25H29ClFN5O4.HCl
      StorageStoreat-20°C
      Purity≥98%(HPLC)
      CASNumber1642187-96-9
      PubChemID86765292
      InChIKeyNUIXGNLBPARAII-UHFFFAOYSA-N
      SmilesO=C(NC(C)C)CN1C(C2=CC(OCCCN3CCOCC3)=CN=C2N=C1C4=CC=C(F)C(Cl)=C4)=O.Cl

      Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

      AllTocrisproductsareintendedforlaboratoryresearchuseonly.

      SolubilityData

      SolventMaxConc.mg/mLMaxConc.mM
      Solubility
      water55.44100
      DMSO55.44100

      PreparingStockSolutions

      Thefollowingdataisbasedontheproductmolecularweight554.44.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

      Concentration/SolventVolume/Mass1mg5mg10mg
      1mM1.8mL9.02mL18.04mL
      5mM0.36mL1.8mL3.61mL
      10mM0.18mL0.9mL1.8mL
      50mM0.04mL0.18mL0.36mL