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Tocris/Eletriptan hydrobromide/3862/50/50 mg

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货号: 3862/50

品牌: Tocris

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Description: Orally active, selective 5-HT_1B/1D agonist

Chemical Name: 3-[[(2R)-1-Methyl-2-pyrrolidinyl]methyl]-5-[2-(phenylsulfonyl)ethyl]-1H-indole hydrobromide

Purity: ≥99% (HPLC)

Biological Activity Technical Data Solubility Calculators Datasheets References

Biological Activity

Orally active, selective 5-HT_1B/1D receptor agonist. Produces a dose-dependent reduction in carotid artery blood flow in vivo. Displays antimigraine activity.

Licensing Information

Sold for research purposes under agreement from Pfizer Inc.

Compound Libraries

Eletriptan hydrobromide is also offered as part of the Tocriscreen Plus and Tocriscreen Library of FDA-Approved Compounds. Find out more about compound libraries available from Tocris.

Technical Data

M. Wt	463.43
Formula	C₂₂H₂₆N₂O₂S.HBr
Storage	Desiccate at RT
Purity	≥99% (HPLC)
CAS Number	177834-92-3
PubChem ID	656631
InChI Key	UTINOWOSWSPFLJ-FSRHSHDFSA-N
Smiles	CN1[C@@H](CC3=CNC2=CC=C(CCS(=O)(C4=CC=CC=C4)=O)C=C23)CCC1.Br

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

All Tocris products are intended for laboratory research use only.

Solubility Data

	Solvent	Max Conc. mg/mL	Max Conc. mM
Solubility
Solubility	DMSO	46.34	100

Preparing Stock Solutions

The following data is based on the product molecular weight 463.43. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	2.16 mL	10.79 mL	21.58 mL
5 mM	0.43 mL	2.16 mL	4.32 mL
10 mM	0.22 mL	1.08 mL	2.16 mL
50 mM	0.04 mL	0.22 mL	0.43 mL

Product Datasheets

Certificate of Analysis / Product Datasheet

Safety Datasheet

References

References are publications that support the products' biological activity.

Napier et al (1999) Characterisation of the 5-HT receptor binding profile of eletriptan and kinetics of [³H]-eletriptan binding at human 5-HT_1B and 5-HT_1D receptors. Eur.J.Pharmacol. 368 259 PMID: 10193663

Gupta et al (2000) The in vivo pharmacological profile of eletriptan (UK-116,044): a potent and novel 5-HT(1B/1D) receptor agonist. Eur.J.Pharmacol. 398 73 PMID: 10856450

Willems et al (1998) Porcine carotid vascular effects of eletriptan (UK-116,044): a new 5-HT_1B/1D receptor agonist with anti-migraine activity. Naunyn-Schmied.Arch.Pharmacol. 358 212 PMID:

Keywords: Eletriptan hydrobromide, supplier, 5-HT1B, 5-HT1D, 5-HT1B/1D, selective, orally, active, agonists, receptors, serotonin, Pfizer, 5-HT1B, Receptors, 5-HT1D, Receptors, 5-HT1B, Receptors, Tocris Bioscience

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