BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences
BiologicalActivity
Potent,orallyactiveCB1/CB2receptoragonistwithlimitedbrainpenetration(EC50valuesare6.1and27.9nMforCB1andCB2receptorsrespectively).DisplaysantihyperalgesicactivityinaratmodelofneuropathicpainwithnoCNSsideeffects.
TechnicalData
M.Wt | 368.47 |
Formula | C26H24O2 |
Storage | StoreatRT |
Purity | ≥99%(HPLC) |
CASNumber | 432047-72-8 |
PubChemID | 9799417 |
InChIKey | RSUMDJRTAFBISX-UHFFFAOYSA-N |
Smiles | O=C(C3=CC=CC4=C3C=CC=C4)C2=CC=C(OCCCCC)C1=CC=CC=C12 |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solvent | MaxConc.mg/mL | MaxConc.mM |
---|
Solubility |
---|
DMSO | 36.85 | 100 |
ethanol | 18.42 | 50 |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight368.47.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
---|
1mM | 2.71mL | 13.57mL | 27.14mL |
5mM | 0.54mL | 2.71mL | 5.43mL |
10mM | 0.27mL | 1.36mL | 2.71mL |
50mM | 0.05mL | 0.27mL | 0.54mL |