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Tocris/WIN 55,212-3 mesylate/2327/10/10 mg
  • Tocris/WIN 55,212-3 mesylate/2327/10/10 mg

Tocris/WIN 55,212-3 mesylate/2327/10/10 mg

价格: ¥1548.00 市场价: 2580.00
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货号: 2327
品牌: Tocris
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    • Description:CB2antagoNIST/CB1partialinverseagonist;enantiomerofWIN55,212-2(Cat.No.1038)
      AlternativeNames:(S)-(-)-WIN55,212
      ChemicalName:[(3S)-2,3-Dihydro-5-methyl-3-(4-morpholinylmethyl)pyrrolo[1,2,3-de]-1,4-benzoxazin-6-yl]-1-naphthalenyl-methanonemonomethanesulfonate
      Purity:≥98%(HPLC)
      BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

      BiologicalActivity

      Novel,lowpotencyCB2receptorsilentantagonistandCB1receptorpartialinverseagonist.CompetitivelyantagonizeseffectsofCP55,940(pA2=6.1)andSR144528(pEC50=5.3)atCB2receptorsandactsasapartialinverseagonistatCB1receptors(pIC50=5.5).DisplaysmodestactivityathumanmelatoninMT1andmuscarinicM4receptors,butisselectiveoverseveralotherGPCRs.

      TechnicalData

      M.Wt522.61
      FormulaC27H26N2O3.CH3SO3H
      StorageStoreat+4°C
      Purity≥98%(HPLC)
      CASNumber131543-25-4
      PubChemID11613341
      InChIKeyFSGCSTPOPBJYSX-BDQAORGHSA-N
      SmilesCS(O)(=O)=O.CC1=C(C(=O)C2=CC=CC3=C2C=CC=C3)C2=CC=CC3=C2N1[C@@H](CN1CCOCC1)CO3

      Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

      AllTocrisproductsareintendedforlaboratoryresearchuseonly.

      SolubilityData

      SolventMaxConc.mg/mLMaxConc.mM
      Solubility
      DMSO52.26100mMwithgentlewarming

      PreparingStockSolutions

      Thefollowingdataisbasedontheproductmolecularweight522.61.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

      Concentration/SolventVolume/Mass1mg5mg10mg
      1mM1.91mL9.57mL19.13mL
      5mM0.38mL1.91mL3.83mL
      10mM0.19mL0.96mL1.91mL
      50mM0.04mL0.19mL0.38mL