BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences
BiologicalActivity
Anandamidemembranetransportinhibitor(IC50=14μM)thatisrelativelymetabolicallystable.DisplayssomeaffinityforCB2receptorsbuthasonlyweakaffinityforCB1receptorsandhasnoactivityatVR1receptorsorFAAH.AnticonvulsiveinvivofollowingsystemicadmiNISTration.
TechnicalData
M.Wt | 370.57 |
Formula | C25H38O2 |
Storage | Desiccateat-20°C |
CASNumber | 97452-63-6 |
PubChemID | 126670 |
InChIKey | MPJURNPNPDQYSY-LEWJYISDSA-N |
Smiles | C=[C@](C)[C@@H]1CCC(C)=C[C@H]1[C@]2=C(O)C=C(C(C)(C)CCCCCC)C=C2O |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
Solubility | Solubleinethanol(suppliedpre-dissolvedinanhydrousethanol,5mg/ml) |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight370.57.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
---|
1mM | 2.7mL | 13.49mL | 26.99mL |
5mM | 0.54mL | 2.7mL | 5.4mL |
10mM | 0.27mL | 1.35mL | 2.7mL |
50mM | 0.05mL | 0.27mL | 0.54mL |